SCHEMBL5336598

SCHEMBL5336598

CC(=O)c1ccc(NS(=O)(=O)c2ccccc2I)nc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 7/20 0.48
HDAC4 P56524 7/20 0.48
HDAC1 Q13547 7/20 0.48
HDAC7 Q8WUI4 7/20 0.48
HDAC2 Q92769 7/20 0.48
HDAC10 Q969S8 7/20 0.48
HDAC11 Q96DB2 7/20 0.48
HDAC8 Q9BY41 7/20 0.48
HDAC6 Q9UBN7 7/20 0.48
HDAC9 Q9UKV0 7/20 0.48
HDAC5 Q9UQL6 7/20 0.48
EDNRA P25101 4/20 0.44
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 1/20 0.43
F10 P00742 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
PKLR P30613 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771765 0.78 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4793078 0.76 HDAC3 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5317017 0.73 HDAC3 (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5315898 0.71 KDM4E (0.64) KDM4EMEN1LMNAKMT2AALDH1A1
SCHEMBL5333429 0.69 HDAC3 (0.64) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL31247494 0.69 TYK2 (0.53)
SCHEMBL12588541 0.68 HCAR3 (0.72) KMT2A
SCHEMBL13064470 0.68 HDAC3 (0.62) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5560379 0.68 POLB (0.65) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5564141 0.68 BRD4 (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007067993-A1 INHIBITORS OF HISTONE DEACETYLASE FOR THE TREATMENT OF DISEASE KALYPSYS, INC. (US) 2007-06-14 WO disclosed