SCHEMBL5338149

SCHEMBL5338149

O=c1[nH]nc(-c2ccccc2I)c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
KDM4E B2RXH2 2/20 0.50
POLB P06746 2/20 0.50
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.50
LMNA P02545 2/20 0.47
TSHR P16473 1/20 0.47
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
MAPK1 P28482 1/20 0.46
PRMT5 O14744 1/20 0.45
ROCK2 O75116 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28988471 0.79 ATM (0.61) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL2230907 0.79 ATM (0.61) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL7892211 0.79 NPSR1 (0.61) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL29710440 0.77 ATM (0.73) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL29870198 0.76 NPSR1 (1.00) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL581143 0.76 NPSR1 (1.00) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL30989583 0.76 ATM (0.56) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL10091947 0.76 ATM (0.60) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL23496942 0.75 ATM (0.59) ATMNPSR1KDM4EPOLBALDH1A1
SCHEMBL30719641 0.75 ATM (0.59) ATMNPSR1KDM4EPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794148-A1 NOVEL PHTHALAZINONE DERIVATIVES, AS AURORA-A KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-06-13 EP disclosed
WO-2006032518-A1 NOVEL PHTHALAZINONE DERIVATIVES, AS AURORA-A KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-30 WO disclosed