SCHEMBL533941

SCHEMBL533941

Cc1cc(C)c(N2CCCC2)c(C)c1NS(=O)(=O)c1cc(Cl)cc(Cl)c1NC(=O)CN(c1c(C)cc(C)c(NCc2ccccc2)c1C)S(=O)(=O)c1cc(Cl)cc(Cl)c1O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACLY P53396 15/20 0.36
THRB P10828 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
MMP13 P45452 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533940 0.87 ACLY (0.42) ACLY
SCHEMBL532928 0.77 ACLY (0.49) ACLYMEN1KMT2AMMP1MMP2
SCHEMBL534027 0.75 ACLY (0.55) ACLY
SCHEMBL532815 0.75 ACLY (0.53) ACLY
SCHEMBL533015 0.74 ACLY (0.54) ACLY
SCHEMBL532997 0.74 ACLY (0.39) ACLYMEN1KMT2A
SCHEMBL14288684 0.72 ACLY (0.53) ACLY
SCHEMBL14288635 0.71 ACLY (0.37) ACLYTHRBKMT2A
SCHEMBL532952 0.69 ACLY (0.51) ACLY
SCHEMBL532966 0.69 KMT2A (0.43) ACLYTHRBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed