SCHEMBL5341890

SCHEMBL5341890

COC1C(O)[C@@H](COS(N)(=O)=O)O[C@H]1n1cnc2c(Cl)ncnc21

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA4 P22748 1/20 0.55
CA9 Q16790 1/20 0.55
TYMP P19971 1/20 0.52
ATG7 O95352 5/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
UBA6 A0AVT1 1/20 0.49
UBA7 P41226 1/20 0.49
NAE1 Q13564 1/20 0.49
UBA3 Q8TBC4 1/20 0.49
SAE1 Q9UBE0 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
ADORA3 P0DMS8 1/20 0.48
TARS1 P26639 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1800307 1.00 CA1 (0.55) CA1CA2CA4CA9TYMP
SCHEMBL12617951 1.00 CA1 (0.55) CA1CA2CA4CA9TYMP
SCHEMBL1797504 0.85 LARS1 (0.49) CA1CA2CA4CA9ATG7
SCHEMBL18630612 0.85 LARS1 (0.49) CA1CA2CA4CA9ATG7
SCHEMBL1796936 0.85 MEN1 (0.65) TYMPMEN1KMT2AADORA3
SCHEMBL6635214 0.85 MEN1 (0.65) TYMPMEN1KMT2AADORA3
SCHEMBL21480367 0.80 TYMP (0.56) TYMPMEN1KMT2AADORA3
SCHEMBL5321913 0.79 ATG7 (0.63) CA1CA2CA4CA9ATG7
SCHEMBL1796966 0.79 ATG7 (0.63) CA1CA2CA4CA9ATG7
SCHEMBL1796531 0.79 RXFP1 (0.69) CA1CA2CA4CA9TYMP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848718-A1 INHIBITORS OF E1 ACTIVATING ENZYMES MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-10-31 EP disclosed
WO-2006084281-A1 INHIBITORS OF E1 ACTIVATING ENZYMES MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-08-10 WO disclosed