SCHEMBL5345562

SCHEMBL5345562

CCCc1nnc(NC(=O)Oc2ccccc2)s1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.67
ALDH1A1 P00352 6/20 0.64
POLB P06746 2/20 0.64
MEN1 O00255 1/20 0.64
MIF P14174 1/20 0.64
KMT2A Q03164 1/20 0.64
RECQL P46063 1/20 0.63
LMNA P02545 3/20 0.61
KDM4E B2RXH2 2/20 0.60
USP2 O75604 1/20 0.60
HPGD P15428 1/20 0.60
HSD17B10 Q99714 1/20 0.60
SMN1; SMN2 Q16637 5/20 0.59
RAB9A P51151 3/20 0.59
GAA P10253 2/20 0.59
NPC1 O15118 2/20 0.59
NPSR1 Q6W5P4 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
TSHR P16473 1/20 0.58
RXFP1 Q9HBX9 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011592 0.91 POLB (0.68) GLSALDH1A1POLBMEN1MIF
SCHEMBL17193491 0.89 GLS (0.82) GLSALDH1A1POLBMEN1MIF
SCHEMBL17193288 0.88 GLS (0.80) GLSALDH1A1POLBMEN1MIF
SCHEMBL17193292 0.86 GLS (0.64) GLSALDH1A1POLBMEN1MIF
SCHEMBL15724893 0.86 GLS (0.67) GLS
SCHEMBL17193290 0.85 GLS (0.65) GLSALDH1A1POLBMEN1MIF
SCHEMBL17193289 0.84 GLS (0.64) GLSALDH1A1POLBMEN1MIF
SCHEMBL14987305 0.81 GLS (1.00) GLS
SCHEMBL17193287 0.81 GLS (0.66) GLSALDH1A1POLBMEN1MIF
SCHEMBL17655086 0.80 GLS (0.98) GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7288537-B2 Azetidine derivatives as CCR-3 receptor antagonists NOVARTIS AG (CH) 2007-10-30 US disclosed
US-20050222118-A1 Azetidine derivatives as ccr-3 receptor antagonists NOVARTIS AG (CH) 2005-10-06 US disclosed
EP-1487435-A1 AZETIDINE DERIVATIVES AS CCR-3 RECEPTOR ANTAGONISTS Novartis AG (CH) 2004-12-22 EP disclosed
WO-2003077907-A1 AZETIDINE DERIVATIVES AS CCR-3 RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2003-09-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050222118-A1 Azetidine derivatives as ccr-3 receptor antagonists CCR3, CCR1, CCR9 GLS 4715/4885ALDH1A1 2840/4885POLB 4233/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.