SCHEMBL534900

SCHEMBL534900

COCc1cc(-c2nc(-c3ccc(CCO)cc3)no2)ccc1-c1ccccc1C.COCc1cc(-c2nc(-c3cccc(CCO)c3)no2)ccc1-c1ccccc1C.COCc1cc(-c2nc(-c3cccc(CO)c3)no2)ccc1-c1ccccc1C

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.61
S1PR3 Q99500 5/20 0.61
NR1H4 Q96RI1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL410830 0.95 S1PR1 (0.67) S1PR1S1PR3NR1H4
SCHEMBL408734 0.93 S1PR1 (0.69) S1PR1S1PR3NR1H4
SCHEMBL410568 0.92 S1PR1 (0.68) S1PR1S1PR3NR1H4
SCHEMBL320407 0.88 S1PR1 (0.70) S1PR1S1PR3NR1H4
SCHEMBL2809467 0.85 S1PR1 (0.64) S1PR1S1PR3NR1H4
SCHEMBL534796 0.85 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL410691 0.85 S1PR1 (0.63) S1PR1S1PR3NR1H4
SCHEMBL410379 0.84 S1PR1 (0.62) S1PR1S1PR3NR1H4
SCHEMBL2806714 0.84 S1PR1 (0.62) S1PR1S1PR3
SCHEMBL2810457 0.83 S1PR1 (0.61) S1PR1S1PR3NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414341-A2 OXADIAZOLE DERIVATIVES Merck Serono SA (CH) 2012-02-08 EP disclosed
WO-2010115751-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed