SCHEMBL5350685

SCHEMBL5350685

CCCc1nccn1CC(=O)c1ncccc1-c1ccc(N2C[C@H](Cn3ccnn3)OC2=O)cc1F

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.59
CYP2D6 P10635 1/20 0.59
MAOA P21397 17/20 0.57
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359994 0.87 CYP3A4 (0.59) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL4896038 0.86 MAOA (0.74) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL4897434 0.81 MAOA (0.75) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL3328495 0.79 CYP3A4 (0.79) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL3328501 0.79 CYP3A4 (0.79) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL3328493 0.79 CYP3A4 (0.79) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL4887794 0.78 MAOA (0.72) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL4895217 0.77 MAOA (0.81) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL4895902 0.75 MAOA (0.74) CYP3A4CYP2D6MAOACYP2C9
SCHEMBL4901157 0.75 MAOA (0.80) CYP3A4CYP2D6MAOACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753754-A1 3- '4- {6-SUBSTITUTED ALKANOYL) PYRIDIN-3-YL} -3-PHENYL! -5- (1H-1, 2, 3-TRIAZOL-1-YLMETHYL) -1, 3-OXAZOLIDIN-2-ONES AS ANTIBACTERIAL AGENTS AstraZeneca AB (SE) 2007-02-21 EP disclosed
WO-2005116022-A1 3- `4- {6-SUBSTITUTED ALKANOYL) PYRIDIN-3-YL} -3-PHENYL! -5- (1H-1, 2, 3-TRIAZOL-1-YLMETHYL) -1, 3-OXAZOLIDIN-2-ONES AS ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2005-12-08 WO disclosed