SCHEMBL5352269

SCHEMBL5352269

COCCOc1ccnc(CSc2nc3ccccc3[nH]2)c1C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.72
NPC1 O15118 5/20 0.72
CYP2C9 P11712 4/20 0.72
CYP1A2 P05177 2/20 0.72
CYP2D6 P10635 2/20 0.72
CYP2C19 P33261 2/20 0.72
CYP3A4 P08684 1/20 0.72
KMT2A Q03164 4/20 0.56
LMNA P02545 4/20 0.56
MAPT P10636 3/20 0.56
DDAH1 O94760 1/20 0.56
ALDH1A1 P00352 1/20 0.56
HTR1A P08908 1/20 0.56
ADORA3 P0DMS8 1/20 0.56
IDE P14735 1/20 0.56
HPGD P15428 1/20 0.56
ADRA2B P18089 1/20 0.56
TBXA2R P21731 1/20 0.56
ACHE P22303 1/20 0.56
PTGS1 P23219 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501939 0.97 RAB9A (0.68) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL1306777 0.95 RAB9A (0.71) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL29538889 0.95 RAB9A (0.71) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL8502308 0.95 RAB9A (0.71) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL5738053 0.94 RAB9A (0.70) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL5738051 0.94 RAB9A (0.70) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL8503121 0.93 RAB9A (0.66) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL13645586 0.93 RAB9A (0.68) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL31515434 0.92 CYP2C9 (0.74) RAB9ANPC1CYP2C9CYP1A2CYP2D6
SCHEMBL8503345 0.91 RAB9A (0.64) RAB9ANPC1CYP2C9CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007129328-A2 PROCESS FOR PREPARING 2-[PYRIDINYL]SULFINYL-SUBSTITUTED BENZIMIDAZOLES CADILA HEALTHCARE LIMITED (IN) 2007-11-15 WO disclosed
WO-2007129328-A2 PROCESS FOR PREPARING 2-[PYRIDINYL]SULFINYL-SUBSTITUTED BENZIMIDAZOLES CADILA HEALTHCARE LIMITED (IN) 2007-11-15 WO disclosed
US-5708013-A BENZIMIDAZOLESULFOXIDE DERIVATIVES EISAI CO., LTD. (JP) 1998-01-13 US disclosed