SCHEMBL5352279

SCHEMBL5352279

CN(C)c1ccc(CNC(=S)[C@@H](CCC2CCCCC2)NC(=O)[C@@H]2CSCN2)cc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
MAPK11 Q15759 1/20 0.35
GAA P10253 2/20 0.35
SRC P12931 1/20 0.35
KCNH2 Q12809 3/20 0.35
DDR1 Q08345 1/20 0.34
DDR2 Q16832 1/20 0.34
BACE1 P56817 1/20 0.34
POLB P06746 2/20 0.33
MC4R P32245 4/20 0.33
MC5R P33032 3/20 0.33
MC3R P41968 1/20 0.33
MC1R Q01726 1/20 0.33
MAPT P10636 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4845539 0.88 ALDH1A1 (0.46) HTR2CSRCPOLBMAPT
SCHEMBL5344813 0.88 ALDH1A1 (0.46) HTR2CSRCPOLBMAPT
Hydrochloric Acid SCHEMBL5363345 0.87 ALDH1A1 (0.45) HTR2CSRCPOLBMAPT
Hydrochloric Acid SCHEMBL5343346 0.87 ALDH1A1 (0.45) HTR2CSRCPOLBMAPT
SCHEMBL4842911 0.85 EPHX1 (0.43) HTR2CHTR2BGAAMAPT
Hydrochloric Acid SCHEMBL5361556 0.85 EPHX1 (0.43) HTR2CHTR2BGAAMAPT
SCHEMBL4843557 0.85 CACNA1B (0.43) MAPK14HTR2CHTR2BMAPK11SRC
Hydrochloric Acid SCHEMBL4841873 0.84 CACNA1B (0.43) MAPK14HTR2CHTR2BMAPK11SRC
SCHEMBL5356917 0.83 MAPK14 (0.40) MAPK14HTR2CHTR2BMAPK11GAA
SCHEMBL5354944 0.83 MAPK14 (0.35) MAPK14HTR2CHTR2BMAPK11GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7166590-B2 Amino acid derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 2007-01-23 US claimed
EP-0997147-B1 AMINO ACID DERIVATIVES ONO PHARMACEUTICAL CO (JP) 2006-03-15 EP claimed
EP-0997147-A1 AMINO ACID DERIVATIVES Ono Pharmaceutical Co., Ltd. (JP) 2000-05-03 EP claimed
EP-0997147-B1 AMINO ACID DERIVATIVES ONO PHARMACEUTICAL CO (JP) 2006-03-15 EP disclosed
EP-0997147-A1 AMINO ACID DERIVATIVES Ono Pharmaceutical Co., Ltd. (JP) 2000-05-03 EP disclosed