SCHEMBL5352528

SCHEMBL5352528

Cc1cccc(C2CC2C(=O)N2CCC(CNc3ncc(F)cn3)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.51
GRIN2B Q13224 10/20 0.50
HRH3 Q9Y5N1 5/20 0.43
HCRTR1 O43613 2/20 0.42
VNN1 O95497 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5351371 0.93 GRIN2B (0.52) SIGMAR1GRIN2BHRH3VNN1
SCHEMBL5352837 0.91 GRIN2B (0.60) SIGMAR1GRIN2B
SCHEMBL5351992 0.88 SIGMAR1 (0.59) SIGMAR1GRIN2BHRH3
SCHEMBL5355769 0.85 GRIN2B (0.60) SIGMAR1GRIN2BHRH3
SCHEMBL5778248 0.84 SIGMAR1 (0.51) SIGMAR1GRIN2BHRH3
SCHEMBL5345695 0.84 SIGMAR1 (0.51) SIGMAR1GRIN2BHRH3
Hydrochloric Acid SCHEMBL5356897 0.83 SIGMAR1 (0.50) SIGMAR1GRIN2BHRH3
SCHEMBL5347589 0.83 SIGMAR1 (0.50) SIGMAR1GRIN2BHRH3HCRTR1VNN1
SCHEMBL5352378 0.83 SIGMAR1 (0.50) SIGMAR1GRIN2BHRH3HCRTR1VNN1
SCHEMBL14502230 0.83 SIGMAR1 (0.50) SIGMAR1GRIN2BHRH3HCRTR1VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217716-B2 N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists MERCK & CO., INC. (US) 2007-05-15 US disclosed
US-7217716-B2 N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists MERCK & CO., INC. (US) 2007-05-15 US disclosed
US-7217716-B2 N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists MERCK & CO., INC. (US) 2007-05-15 US disclosed
US-7053089-B2 N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists MERCK & CO., INC. (US) 2006-05-30 US disclosed
EP-1379520-B1 N-SUBSTITUTED NONARYL-HETEROCYCLIC NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2006-04-26 EP disclosed