SCHEMBL5354295

SCHEMBL5354295

Cc1ccc(Nc2ncnc3oc(-c4ccc(N)cc4)cc23)cc1O

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.52
RAF1 P04049 1/20 0.52
KDR P35968 9/20 0.49
RET P07949 1/20 0.49
KIF5B P33176 1/20 0.49
EGFR P00533 10/20 0.46
GSK3B P49841 6/20 0.46
FLT1 P17948 1/20 0.43
FLT4 P35916 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5358888 0.86 BRAF (0.59) BRAFRAF1KDRRETKIF5B
SCHEMBL5362131 0.86 ALK (0.45) BRAFRAF1KDRRETKIF5B
SCHEMBL5355580 0.80 AHR (0.52) BRAFRAF1KDRRETEGFR
SCHEMBL14355897 0.78 EGFR (0.52) KDREGFRGSK3B
SCHEMBL5355467 0.77 EGFR (0.58) RAF1KDREGFRGSK3B
SCHEMBL5358390 0.73 ABCG2 (0.53) BRAFRAF1KDRRETKIF5B
SCHEMBL5357333 0.70 RAF1 (0.48) BRAFRAF1KDREGFRGSK3B
SCHEMBL6417988 0.69 GSK3B (0.57) KDREGFRGSK3B
SCHEMBL5564873 0.69 KDR (0.55) BRAFRAF1KDRRETKIF5B
SCHEMBL5559096 0.69 BRAF (0.53) BRAFRAF1KDRRETKIF5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294633-B2 Oxazolo-and furopyrimidines and their use in medicaments against tumors NOVARTIS AG (CH) 2007-11-13 US claimed
EP-1390371-B1 OXAZOLO-AND FUROPYRIMIDINES AND THEIR USE IN MEDICAMENTS AGAINST TUMORS NOVARTIS AG (CH) 2006-03-08 EP claimed
US-20040152892-A1 Oxazolo-and furopyrimidines and their use in medicaments against tumors NOVARTIS AG (CH) 2004-08-05 US claimed
EP-1390371-A1 OXAZOLO-AND FUROPYRIMIDINES AND THEIR USE IN MEDICAMENTS AGAINST TUMORS Novartis AG (CH) 2004-02-25 EP claimed
WO-2002092603-A1 OXAZOLO-AND FUROPYRIMIDINES AND THEIR USE IN MEDICAMENTS AGAINST TUMORS NOVARTIS AG (CH) 2002-11-21 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040152892-A1 Oxazolo-and furopyrimidines and their use in medicaments against tumors DPYD, COXFA4L2, MSH2 BRAF 657/4885RAF1 2306/4885KDR 2394/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.