SCHEMBL535511

SCHEMBL535511

CCCCOC(=O)N1CCC(c2ccn(C)c(=O)c2)C(c2ccc(-c3ccccc3CCNC(C)=O)cc2Cl)C1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
REN P00797 15/20 0.66
KCNH2 Q12809 12/20 0.66
CYP3A4 P08684 1/20 0.48
MTNR1A P48039 2/20 0.33
MTNR1B P49286 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533878 0.90 REN (0.54) RENKCNH2CYP3A4
SCHEMBL556870 0.84 REN (0.75) RENKCNH2CYP3A4PTGDR2
SCHEMBL535144 0.83 REN (0.74) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL534449 0.81 REN (0.66) RENKCNH2CYP3A4PTGDR2
SCHEMBL556618 0.81 REN (0.75) RENKCNH2CYP3A4PTGDR2
SCHEMBL556921 0.80 REN (1.00) RENKCNH2CYP3A4
SCHEMBL556726 0.80 REN (1.00) RENKCNH2CYP3A4
SCHEMBL557684 0.80 REN (0.61) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL556463 0.79 REN (0.58) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL534057 0.78 REN (0.58) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed