SCHEMBL5357658

SCHEMBL5357658

O=c1[nH]c2cc(F)ccc2cc1-c1cc2cc(S(=O)(=O)N3CCNCC3)ccc2[nH]1

nearest known ligand 0.78

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.78
TDO2 P48775 6/20 0.48
PKM P14618 1/20 0.47
RXFP1 Q9HBX9 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CHEK1 O14757 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367396 0.88 KDR (1.00) KDRPKMMEN1KMT2AKDM4E
SCHEMBL5357068 0.85 KDR (0.88) KDRPKMMEN1KMT2AKDM4E
SCHEMBL5356996 0.84 KDR (0.79) KDRPKMMEN1KMT2AKDM4E
SCHEMBL5355012 0.76 KDR (1.00) KDRPKMMEN1KMT2AKDM4E
SCHEMBL19126788 0.76 KDR (0.55) KDRTDO2PKMRXFP1MEN1
SCHEMBL30810537 0.76 KDR (0.55) KDRTDO2PKMRXFP1MEN1
SCHEMBL5357342 0.76 KDR (0.74) KDRPKMCHEK1
SCHEMBL14590416 0.74 KDR (0.88) KDRPKMMEN1KMT2AKDM4E
SCHEMBL5371286 0.73 KDR (0.79) KDRMEN1KMT2AKDM4E
SCHEMBL5370747 0.73 KDR (0.67) KDRTDO2PKMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed