SCHEMBL5370747

SCHEMBL5370747

O=c1[nH]c2ccccc2cc1-c1[nH]c2ccc(S(=O)(=O)N3CCNCC3)cc2c1F

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.67
PKM P14618 2/20 0.49
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
BLM P54132 1/20 0.41
TDO2 P48775 2/20 0.41
GAA P10253 2/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ERBB2 P04626 1/20 0.39
PTK6 Q13882 1/20 0.39
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5352066 0.92 KDR (0.64) KDRPKMTDP1KDM4EALDH1A1
SCHEMBL5355475 0.89 KDR (0.68) KDRPKMTDP1KDM4EALDH1A1
SCHEMBL5362580 0.84 KDR (0.70) KDRPKMTDP1KDM4EALDH1A1
SCHEMBL5362476 0.82 KDR (0.65) KDRPKMTDP1KDM4EALDH1A1
SCHEMBL5367396 0.81 KDR (1.00) KDRPKMKDM4EALDH1A1MEN1
SCHEMBL5357068 0.79 KDR (0.88) KDRPKMTDP1KDM4EALDH1A1
SCHEMBL14559410 0.77 KDR (0.57) KDRKDM4EALDH1A1LMNAMEN1
SCHEMBL5359215 0.77 KDR (0.67) KDRTDP1KDM4EALDH1A1LMNA
SCHEMBL5371327 0.76 SLC6A2 (0.56) KDRKDM4EALDH1A1TSHRHSD17B10
SCHEMBL5367711 0.74 KDR (0.70) KDRPKMKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed