SCHEMBL5357992

SCHEMBL5357992

CN(C)/C=C(\C(=O)c1ccc(F)cc1)c1ccnc(NC(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 1/20 0.39
CYP17A1 P05093 3/20 0.38
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RIPK3 Q9Y572 1/20 0.36
AR P10275 1/20 0.35
GSK3B P49841 5/20 0.35
KCNQ4 P56696 1/20 0.35
KCNQ5 Q9NR82 1/20 0.35
MAPT P10636 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
ATR Q13535 1/20 0.34
GSK3A P49840 2/20 0.34
PIK3C3 Q8NEB9 1/20 0.34
IGF1R P08069 1/20 0.34
RORC P51449 2/20 0.34
DYRK1A Q13627 1/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5357995 1.00 HTR1F (0.39) HTR1FCYP17A1NPC1TP53RAB9A
SCHEMBL5356752 0.90 CYP17A1 (0.39) CYP17A1GSK3BAAK1ATRGSK3A
SCHEMBL5356757 0.90 CYP17A1 (0.39) CYP17A1GSK3BAAK1ATRGSK3A
SCHEMBL5348564 0.90 CYP11B1 (0.40) CYP17A1NPC1RAB9ASMN1; SMN2AAK1
SCHEMBL5348562 0.90 CYP11B1 (0.40) CYP17A1NPC1RAB9ASMN1; SMN2AAK1
SCHEMBL5351318 0.90 ACACB (0.39) CYP17A1NPC1RAB9AGSK3BAAK1
SCHEMBL5351320 0.90 ACACB (0.39) CYP17A1NPC1RAB9AGSK3BAAK1
SCHEMBL5355228 0.89 NPC1 (0.37) CYP17A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL5355226 0.89 NPC1 (0.37) CYP17A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL5348696 0.85 CYP11B1 (0.38) CYP17A1GSK3BMAPTAAK1ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1553096-B1 PYRAZOLE COMPOUNDS UBE INDUSTRIES (JP) 2012-10-31 EP disclosed
US-7294625-B2 Pyrazole compounds UBE INDUSTRIES, LTD. (JP) 2007-11-13 US disclosed
US-20060063934-A1 3-Pyridazonyl- or triazolopyridazinyl- 4-pyridinyl- or pyrimidinyl- pyrazoles, e.g., 4-(2-aminopyridin-4-yl)-3-phenyl-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazole; p38MAP kinase inhibitors, used to treat rheumatoid arthritis UBE INDUSTRIES, LTD. (JP) 2006-03-23 US disclosed
EP-1553096-A1 PYRAZOLE COMPOUNDS Ube Industries, Ltd. (JP) 2005-07-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063934-A1 3-Pyridazonyl- or triazolopyridazinyl- 4-pyridinyl- or pyrimidinyl- pyrazoles, e.g., 4-(2-aminopyridin-4-yl)-3-phenyl-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazole; p38MAP kinase inhibitors, used to treat rheumatoid arthritis CNKSR1, MAPK1, MAPK3 HTR1F 881/4885CYP17A1 4123/4885NPC1 4466/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.