SCHEMBL5358909

SCHEMBL5358909

CC#CCn1c(Br)nc2cnn(Cc3ccc4ncccc4n3)c(=O)c21

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 19/20 0.43
CHRM1 P11229 5/20 0.43
FAP Q12884 2/20 0.37
CYP3A4 P08684 1/20 0.33
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362704 0.83 DPP4 (0.64) DPP4CHRM1FAP
SCHEMBL5362379 0.83 DPP4 (0.41) DPP4CHRM1FAP
SCHEMBL4249672 0.83 DPP4 (0.44) DPP4CHRM1FAPCYP3A4
SCHEMBL4252373 0.81 DPP4 (0.45) DPP4CHRM1FAPCYP3A4
SCHEMBL5359347 0.81 DPP4 (0.42) DPP4CHRM1FAPCYP3A4
SCHEMBL5361062 0.81 DPP4 (0.66) DPP4CHRM1FAP
SCHEMBL3917633 0.79 DPP4 (0.54) DPP4CHRM1FAPCYP3A4
SCHEMBL4070957 0.79 DPP4 (0.68) DPP4CHRM1
SCHEMBL4069497 0.79 DPP4 (0.68) DPP4CHRM1
SCHEMBL3207468 0.76 DPP4 (0.71) DPP4CHRM1FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217711-B2 Piperazin-1-yl and 2-([1,4]diazepan-1-yl)-imidazo[4,5-d]-pyridazin-4-ones, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-15 US disclosed