SCHEMBL5362379

SCHEMBL5362379

CC#CCn1c(Br)nc2cnn(Cc3ccc4nccnc4c3)c(=O)c21

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 16/20 0.41
CHRM1 P11229 5/20 0.41
FAP Q12884 1/20 0.33
PKM P14618 1/20 0.32
PKLR P30613 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366056 0.87 DPP4 (0.40) DPP4CHRM1FAPPKMPKLR
SCHEMBL5358438 0.84 DPP4 (0.39) DPP4CHRM1FAPPKMPKLR
SCHEMBL5370066 0.83 DPP4 (0.62) DPP4CHRM1FAP
SCHEMBL5358909 0.83 DPP4 (0.43) DPP4CHRM1FAP
SCHEMBL4248894 0.81 DPP4 (0.43) DPP4CHRM1
SCHEMBL5359347 0.80 DPP4 (0.42) DPP4CHRM1FAP
SCHEMBL5365295 0.79 DPP4 (0.41) DPP4CHRM1ALDH1A1
SCHEMBL3975290 0.78 DPP4 (0.50) DPP4CHRM1FAPPKMALDH1A1
SCHEMBL1069921 0.78 DPP4 (0.68) DPP4CHRM1
SCHEMBL8278518 0.78 DPP4 (0.68) DPP4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217711-B2 Piperazin-1-yl and 2-([1,4]diazepan-1-yl)-imidazo[4,5-d]-pyridazin-4-ones, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-15 US disclosed