SCHEMBL5358920

SCHEMBL5358920

O=C(NCC1CN(C(=O)OCCc2ccccc2)CCO1)c1ccc(O)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
HPGD P15428 3/20 0.44
ENPP2 Q13822 1/20 0.43
GRIN2B Q13224 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NAMPT P43490 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425436 0.91 MEN1 (0.50) DRD2DRD4DRD3HPGDENPP2
SCHEMBL14425317 0.91 MEN1 (0.50) DRD2DRD4DRD3HPGDENPP2
SCHEMBL5368740 0.91 MEN1 (0.50) DRD2DRD4DRD3HPGDENPP2
SCHEMBL14425361 0.86 F2 (0.46) HPGDENPP2MEN1KMT2AGAA
SCHEMBL5366862 0.86 F2 (0.46) HPGDENPP2MEN1KMT2AGAA
SCHEMBL14425362 0.85 HPGD (0.52) HPGDENPP2MEN1KMT2AGAA
SCHEMBL5364667 0.85 HPGD (0.52) HPGDENPP2MEN1KMT2AGAA
SCHEMBL5370278 0.85 FKBP1A (0.49) DRD2DRD4DRD3HPGDMEN1
SCHEMBL14425318 0.85 FKBP1A (0.49) DRD2DRD4DRD3HPGDMEN1
SCHEMBL5359420 0.83 GRIN2B (0.46) HPGDENPP2GRIN2BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed