SCHEMBL5359891

SCHEMBL5359891

O=C(NCC1CCN(C(=O)OC2Cc3ccccc3C2)CC1)c1ccc(O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.61
TPSAB1 Q15661 5/20 0.60
F2 P00734 4/20 0.60
PRSS1 P07477 4/20 0.60
PRSS2 P07478 4/20 0.60
PRSS3 P35030 4/20 0.60
TPSD1 Q9BZJ3 4/20 0.60
TPSG1 Q9NRR2 4/20 0.60
PLG P00747 2/20 0.60
KDM4E B2RXH2 1/20 0.58
PKM P14618 1/20 0.58
NAMPT P43490 5/20 0.49
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366605 0.88 GRIN2B (0.66) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5371163 0.87 GRIN2B (0.61) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5360921 0.84 GRIN2B (0.60) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5366681 0.84 GRIN2B (0.58) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5378251 0.81 GRIN2B (0.59) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5370671 0.81 NAMPT (0.44) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5370580 0.80 KMT2A (0.58) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5368103 0.80 TPSAB1 (0.71) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5375092 0.79 GRIN2B (0.62) GRIN2BTPSAB1F2PRSS1PRSS2
SCHEMBL5368503 0.79 GRIN2B (0.61) GRIN2BTPSAB1F2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed