SCHEMBL5360124

SCHEMBL5360124

CCOC(=O)c1nn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.50
RAB9A P51151 2/20 0.50
ALDH1A1 P00352 6/20 0.45
ELANE P08246 5/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 2/20 0.45
HPGD P15428 1/20 0.45
TP53 P04637 1/20 0.45
ALOX12 P18054 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
NPSR1 Q6W5P4 2/20 0.44
GLA P06280 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GABRA2 P47869 1/20 0.43
GABRB2 P47870 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19716281 0.87 NPC1 (0.48) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL3076334 0.86 NPC1 (0.47) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL3082411 0.85 NPC1 (0.46) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL3083355 0.85 NPC1 (0.46) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL5363475 0.84 KDM4E (0.48) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL19730343 0.79 UCHL1 (0.42) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL4376014 0.78 TSHR (0.45) NPC1RAB9AALDH1A1HSD17B10KDM4E
SCHEMBL19277273 0.77 NPC1 (0.43) NPC1RAB9AALDH1A1ELANEKDM4E
SCHEMBL23496544 0.77 NPC1 (0.48) NPC1RAB9AALDH1A1ELANEHSD17B10
SCHEMBL1562700 0.77 MAPT (0.45) NPC1RAB9AALDH1A1ELANEHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed