SCHEMBL536037

SCHEMBL536037

COC(=O)c1cc(C)cc(NC(=O)C2(CO[Si](C)(C)C(C)(C)C)C(F)=C(F)C(c3ccccc3)C(F)=C2F)c1N

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
CACNA1F O60840 1/20 0.32
CACNA1D Q01668 1/20 0.32
CACNA1S Q13698 1/20 0.32
CACNA1C Q13936 1/20 0.32
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 2/20 0.30
LMNA P02545 1/20 0.30
RAB9A P51151 1/20 0.30
SIRT3 Q9NTG7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL505290 0.69 HTT (0.36) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL536038 0.66 MEN1 (0.31) ALDH1A1MAPTHPGDKMT2A
SCHEMBL6118859 0.60 KDM4E (0.49) KDM4EALDH1A1MAPTHPGDPOLB
SCHEMBL6118855 0.59 KDM4E (0.55) KDM4EALDH1A1MAPTHPGDPOLB
SCHEMBL9430926 0.59 ALDH1A1 (0.49) KDM4EALDH1A1MAPTHPGDKMT2A
SCHEMBL25591913 0.58 ALDH1A1 (0.50) KDM4EALDH1A1HTTPOLBKMT2A
SCHEMBL12731290 0.57 KDM4E (0.43) KDM4EALDH1A1MAPTHPGDPOLB
SCHEMBL6472720 0.57 KDM4E (0.43) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL30630386 0.56 MRGPRX4 (0.50) KDM4EALDH1A1HTTPOLBKMT2A
SCHEMBL29100989 0.56 MRGPRX4 (0.50) KDM4EALDH1A1HTTPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414328-A2 DIHYDROOROTATE DEHYDROGENASE INHIBITORS Merck Serono S.A. (CH) 2012-02-08 EP disclosed
WO-2010115736-A2 DIHYDROOROTATE DEHYDROGENASE INHIBITORS MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed