SCHEMBL5362152

SCHEMBL5362152

O=C1Nc2ccc(S(=O)(=O)Nc3ccc(C(F)(F)F)cc3)cc2C1=Cc1cc(Cl)ccc1O

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MOGAT2 Q3SYC2 1/20 0.52
MGAT2 Q10469 5/20 0.49
LRRK2 Q5S007 6/20 0.46
PSEN1 P49768 2/20 0.44
PSEN2 P49810 2/20 0.44
APH1B Q8WW43 2/20 0.44
NCSTN Q92542 2/20 0.44
APH1A Q96BI3 2/20 0.44
PSENEN Q9NZ42 2/20 0.44
MGAT1 P26572 1/20 0.43
MGAT3 Q09327 1/20 0.43
PKM P14618 1/20 0.42
TLK2 Q86UE8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5357716 0.91 MOGAT2 (0.54) MOGAT2MGAT2TLK2
SCHEMBL5369245 0.89 MOGAT2 (0.52) MOGAT2MGAT2LRRK2TLK2
SCHEMBL5358023 0.89 MOGAT2 (0.52) MOGAT2MGAT2LRRK2PSEN1PSEN2
SCHEMBL7138959 0.89 MOGAT2 (0.54) MOGAT2MGAT2LRRK2PSEN1PSEN2
SCHEMBL5361507 0.88 MOGAT2 (0.55) MOGAT2MGAT2PKMTLK2
SCHEMBL5358529 0.88 MOGAT2 (0.51) MOGAT2MGAT2LRRK2PSEN1PSEN2
SCHEMBL5367671 0.87 MOGAT2 (0.54) MOGAT2MGAT2PKMTLK2
SCHEMBL5358480 0.87 MOGAT2 (0.52) MOGAT2MGAT2TLK2
SCHEMBL5361643 0.87 MOGAT2 (0.52) MOGAT2MGAT2MGAT1
SCHEMBL7133813 0.86 MOGAT2 (0.52) MOGAT2MGAT2LRRK2PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK MOGAT2 1159/4885MGAT2 4714/4885LRRK2 289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.