SCHEMBL5362853

SCHEMBL5362853

Cn1cc(Cl)c(C=C2C(=O)Nc3ccc(CCCl)cc32)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 2/20 0.40
PSEN1 P49768 5/20 0.39
PSEN2 P49810 5/20 0.39
APH1B Q8WW43 5/20 0.39
NCSTN Q92542 5/20 0.39
APH1A Q96BI3 5/20 0.39
PSENEN Q9NZ42 5/20 0.39
PDPK1 O15530 1/20 0.39
CDK1 P06493 2/20 0.39
CCNB1 P14635 2/20 0.39
LRRK2 Q5S007 4/20 0.38
GSK3B P49841 1/20 0.38
RET P07949 1/20 0.37
PDGFRB P09619 1/20 0.36
NTRK1 P04629 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370004 0.82 MAPT (0.50) NEK2PSEN1PSEN2APH1BNCSTN
SCHEMBL5999800 0.79 GSK3B (0.58) CDK1CCNB1GSK3BPDGFRBNTRK1
SCHEMBL5999807 0.79 GSK3B (0.58) CDK1CCNB1GSK3BPDGFRBNTRK1
SCHEMBL5359158 0.77 SYK (0.53) PDGFRBNTRK1
SCHEMBL5377180 0.76 MEN1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5361124 0.76 KDR (0.64) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5361467 0.75 MEN1 (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7136387 0.75 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7139603 0.75 MEN1 (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7140932 0.75 PSEN1 (0.62) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK NEK2 305/4885PSEN1 3695/4885PSEN2 3641/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.