SCHEMBL5363073

SCHEMBL5363073

CCOC(=O)c1c(C)[nH]c(C=C2C(=O)Nc3ccc(CN)cc32)c1C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 4/20 0.71
FGFR1 P11362 3/20 0.71
ALK Q9UM73 2/20 0.71
RET P07949 2/20 0.71
FLT3 P36888 2/20 0.71
ABL1 P00519 1/20 0.71
PRKAA1 Q13131 12/20 0.55
PRKAA2 P54646 10/20 0.55
LRRK2 Q5S007 1/20 0.54
KDR P35968 8/20 0.54
TLK2 Q86UE8 1/20 0.52
CSF1R P07333 2/20 0.51
PLK4 O00444 1/20 0.50
DCLK1 O15075 1/20 0.50
PDPK1 O15530 1/20 0.50
DAPK3 O43293 1/20 0.50
DYRK3 O43781 1/20 0.50
ROCK2 O75116 1/20 0.50
RPS6KA5 O75582 1/20 0.50
RPS6KA4 O75676 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5363167 0.89 PDGFRB (0.69) PDGFRBFGFR1ALKRETFLT3
SCHEMBL31727096 0.88 PDGFRB (0.74) PDGFRBFGFR1ALKRETFLT3
SCHEMBL19255670 0.88 PDGFRB (0.77) PDGFRBFGFR1ALKRETFLT3
SCHEMBL5373629 0.87 PDGFRB (0.76) PDGFRBFGFR1ALKRETFLT3
SCHEMBL5567713 0.86 ALK (0.76) PDGFRBFGFR1ALKRETFLT3
SCHEMBL31726848 0.86 PDGFRB (0.74) PDGFRBFGFR1ALKRETFLT3
SCHEMBL5392303 0.86 PDGFRB (0.74) PDGFRBFGFR1ALKRETFLT3
SCHEMBL5376617 0.86 PDGFRB (0.74) PDGFRBFGFR1ALKRETFLT3
SCHEMBL5361463 0.85 FGFR1 (0.69) PDGFRBFGFR1ALKRETFLT3
SCHEMBL5365610 0.85 PDGFRB (0.69) PDGFRBFGFR1ALKRETFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK PDGFRB 52/4885FGFR1 112/4885ALK 325/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.