SCHEMBL5364339

SCHEMBL5364339

Fc1ccc2c(c1)CCN2C[CH]COCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.42
MGAT2 Q10469 1/20 0.41
ALOX5 P09917 2/20 0.40
EPHX2 P34913 2/20 0.40
CTSL P07711 5/20 0.40
CTSS P25774 4/20 0.40
CTSK P43235 3/20 0.40
NOTUM Q6P988 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
KDM4A O75164 1/20 0.35
KDM2B Q8NHM5 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27667528 0.77 CTSS (0.48) GRM5MGAT2ALOX5EPHX2CTSL
SCHEMBL3012389 0.77 CTSS (0.48) GRM5MGAT2ALOX5EPHX2CTSL
SCHEMBL5363803 0.72 GRM5 (0.43) GRM5
SCHEMBL5352211 0.70 NOTUM (0.45) MGAT2ALOX5EPHX2CTSLCTSS
SCHEMBL5363794 0.69 NOTUM (0.44) MGAT2ALOX5EPHX2CTSLCTSS
SCHEMBL24823574 0.67 NOTUM (0.49) MGAT2ALOX5EPHX2NOTUMKDM4A
SCHEMBL12060492 0.67 NOTUM (0.53) MGAT2ALOX5EPHX2NOTUMKDM4A
SCHEMBL4572948 0.67 NOTUM (0.50) ALOX5EPHX2CTSLCTSSCTSK
SCHEMBL24495180 0.67 HDAC1 (0.49) ALOX5EPHX2NOTUMKDM4AKDM2B
SCHEMBL29713576 0.67 HDAC1 (0.49) ALOX5EPHX2NOTUMKDM4AKDM2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7307095-B2 Osteoporosis; antiarthritic agents; antidiabetic agents; antiinflammatory agents; Alzheimer's disease; shock; central nervous stsrem disorders; anticancer agents; multiple sclerosis, (S)-2-(Benzooxazol-2-ylamino)-3-cyclohexyl-N-[2-(5-fluoro-2,3-dihydro-indol-1-yl)-ethyl]-propionamide IRM LLC (BM) 2007-12-11 US disclosed