SCHEMBL5364632

SCHEMBL5364632

Cc1ccc(Cc2cc(C)c(=O)[nH]n2)cc1Oc1cccc(C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
FNTA P49354 2/20 0.40
FNTB P49356 2/20 0.40
PGGT1B P53609 2/20 0.40
P2RX3 P56373 4/20 0.37
PIK3R1 P27986 3/20 0.37
PIK3CA P42336 3/20 0.37
EPAS1 Q99814 1/20 0.37
AR P10275 1/20 0.36
NOD1 Q9Y239 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
LRRK2 Q5S007 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14570769 0.91 CYP3A4 (0.53) CYP3A4CYP2C9CYP2C19PRMT5WDR77
SCHEMBL5375295 0.88 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19PRMT5WDR77
SCHEMBL5365473 0.86 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19EPAS1
SCHEMBL5375470 0.82 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19PIK3R1PIK3CA
SCHEMBL4809760 0.81 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19PRMT5WDR77
SCHEMBL5369098 0.79 CYP3A4 (0.57) CYP3A4CYP2C9CYP2C19P2RX3PIK3R1
SCHEMBL5370521 0.79 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19PRMT5WDR77
SCHEMBL14570768 0.79 CYP3A4 (0.57) CYP3A4CYP2C9CYP2C19PIK3R1PIK3CA
SCHEMBL5419846 0.79 CYP3A4 (0.53) CYP3A4CYP2C9CYP2C19PIK3R1PIK3CA
SCHEMBL5421566 0.79 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19PIK3R1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed