SCHEMBL5364969

SCHEMBL5364969

O=C(O)c1cc(F)c(F)cc1Oc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.45
PTGER2 P43116 1/20 0.45
XDH P47989 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PNLIP P16233 1/20 0.43
KDM4E B2RXH2 1/20 0.43
POLB P06746 1/20 0.43
DHODH Q02127 1/20 0.42
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21274769 0.88 PNLIP (0.45) PTGER4PTGER2XDHPNLIPDHODH
SCHEMBL4445272 0.84 PTGER4 (0.59) PTGER4PTGER2XDHPNLIPKDM4E
SCHEMBL4450925 0.84 PTGER4 (0.49) PTGER4PTGER2XDHKDM4EDHODH
SCHEMBL22319389 0.80 PTGER4 (0.49) PTGER4PTGER2XDHKDM4EPOLB
SCHEMBL31028181 0.80 PTGER4 (0.49) PTGER4PTGER2XDHKDM4EPOLB
SCHEMBL22334429 0.80 DHODH (0.42) PTGER4PTGER2XDHKDM4EPOLB
SCHEMBL21274598 0.80 KDM4E (0.50) KDM4EPOLB
SCHEMBL11578048 0.79 KDM4E (0.50) PTGER4PTGER2SLC6A2SLC6A4SLC6A3
SCHEMBL8282850 0.79 PTGER4 (0.48) PTGER4PTGER2XDHPNLIPKDM4E
SCHEMBL4448975 0.79 PTGER4 (0.62) PTGER4PTGER2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663979-B1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS RAQUALIA PHARMA INC (JP) 2013-10-09 EP disclosed
US-7238714-B2 Aryl or heteroaryl amide compounds PFIZER JAPAN, INC. (JP) 2007-07-03 US disclosed
EP-1663979-A1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS PFIZER INC. (US) 2006-06-07 EP disclosed
US-20050065188-A1 Aryl or heteroaryl amide compounds ASKAT INC. (JP) 2005-03-24 US disclosed
WO-2005021508-A1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS PFIZER INC. (US) 2005-03-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065188-A1 Aryl or heteroaryl amide compounds HRH2, PTGER1, LTB4R2 PTGER4 13/4885PTGER2 11/4885XDH 877/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.