SCHEMBL5365162

SCHEMBL5365162

O=C1Nc2ccc(CCCl)cc2C1=Cc1cc2ccccc2nc1Cl

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.48
LRRK2 Q5S007 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RPS6KA3 P51812 2/20 0.41
PDPK1 O15530 1/20 0.40
FLT3 P36888 3/20 0.39
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
ALK Q9UM73 1/20 0.39
MAP3K7 O43318 1/20 0.39
TAB1 Q15750 1/20 0.39
MDM2 Q00987 2/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7132958 0.83 PDGFRB (0.43) GSK3BLRRK2MEN1KMT2ARPS6KA3
SCHEMBL7137938 0.82 LRRK2 (0.46) GSK3BLRRK2RPS6KA3PDPK1MAOA
SCHEMBL7139603 0.81 MEN1 (0.49) GSK3BLRRK2MEN1KMT2ARPS6KA3
SCHEMBL7134805 0.79 CHEK1 (0.42) GSK3BLRRK2MEN1KMT2ARPS6KA3
SCHEMBL7136594 0.78 NPC1 (0.62) GSK3BLRRK2MEN1KMT2ARPS6KA3
SCHEMBL7139419 0.78 MEN1 (0.67) GSK3BLRRK2MEN1KMT2ARPS6KA3
SCHEMBL7135626 0.78 MDM2 (0.50) LRRK2RPS6KA3MDM2PSEN1PSEN2
SCHEMBL5361803 0.77 LRRK2 (0.65) LRRK2PDPK1FLT3MAOAMAOB
SCHEMBL5370088 0.77 SRC (0.51) GSK3BLRRK2MEN1KMT2APDPK1
SCHEMBL5366450 0.76 FLT3 (0.50) LRRK2MEN1KMT2ARPS6KA3FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK GSK3B 315/4885LRRK2 289/4885MEN1 3855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.