SCHEMBL5365366

SCHEMBL5365366

N#Cc1cc(F)cc(Oc2cc(Cc3ccc(=O)[nH]n3)ccc2Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
EPAS1 Q99814 14/20 0.40
VEGFA P15692 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377805 0.93 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19
SCHEMBL5382537 0.90 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19EPAS1VEGFA
SCHEMBL5381993 0.90 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19EPAS1VEGFA
SCHEMBL5385784 0.88 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19EPAS1VEGFA
SCHEMBL14559745 0.88 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19EPAS1VEGFA
SCHEMBL5377332 0.88 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19EPAS1VEGFA
SCHEMBL14559716 0.87 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19EPAS1VEGFA
SCHEMBL5386135 0.87 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19
SCHEMBL5377579 0.86 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19EPAS1
SCHEMBL5385097 0.86 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19EPAS1VEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed