SCHEMBL5377579

SCHEMBL5377579

N#Cc1cccc(Oc2cc(Cc3ccc(=O)[nH]n3)ccc2Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.52
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
PGGT1B P53609 1/20 0.40
P2RX3 P56373 4/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
EPAS1 Q99814 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
DRD4 P21917 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
ERBB3 P21860 1/20 0.36
ERBB4 Q15303 1/20 0.36
HTR2A P28223 2/20 0.36
KCNH2 Q12809 2/20 0.36
SLC6A4 P31645 1/20 0.36
CYP19A1 P11511 1/20 0.35
NR1H4 Q96RI1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377805 0.91 CYP3A4 (0.45) CYP3A4FNTAFNTBPGGT1BCYP2C9
SCHEMBL5386135 0.89 CYP3A4 (0.45) CYP3A4PRMT5WDR77CYP2C9CYP2C19
SCHEMBL5370850 0.88 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19HTR2AKCNH2
SCHEMBL5382537 0.88 CYP3A4 (0.47) CYP3A4EPAS1CYP2C9CYP2C19HTR2A
SCHEMBL5374410 0.88 CYP3A4 (0.49) CYP3A4FNTAFNTBPGGT1BP2RX3
SCHEMBL5375295 0.88 CYP3A4 (0.47) CYP3A4FNTAFNTBPGGT1BP2RX3
SCHEMBL5370328 0.88 CYP3A4 (0.47) CYP3A4FNTAFNTBPGGT1BP2RX3
SCHEMBL5370543 0.87 CYP3A4 (0.46) CYP3A4FNTAFNTBPGGT1BP2RX3
SCHEMBL5365181 0.86 CYP3A4 (0.67) CYP3A4FNTAFNTBPGGT1BPRMT5
SCHEMBL5365366 0.86 CYP3A4 (0.51) CYP3A4EPAS1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed