SCHEMBL5365892

SCHEMBL5365892

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1cn[nH]c1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.65
ROCK2 O75116 2/20 0.40
CYP11B2 P19099 4/20 0.39
CYP11B1 P15538 2/20 0.37
PDE9A O76083 1/20 0.37
PDE1C Q14123 1/20 0.37
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
NAMPT P43490 1/20 0.36
CYP19A1 P11511 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468889 0.83 AR (0.86) ARCYP11B2CYP11B1PDE9APDE1C
SCHEMBL6464451 0.80 AR (0.80) ARCYP11B2CYP11B1CCNCCDK8
SCHEMBL24411088 0.80 AR (0.76) ARCYP11B2CYP11B1PDE9APDE1C
SCHEMBL6465872 0.80 AR (0.76) ARCYP11B2CYP11B1PDE9APDE1C
SCHEMBL24414502 0.79 AR (0.80) ARCYP11B2CYP11B1PDE9APDE1C
SCHEMBL6464131 0.79 AR (0.80) ARCYP11B2CYP11B1CYP19A1GRIN1
SCHEMBL6465272 0.78 AR (1.00) ARCYP11B2CYP11B1PDE9APDE1C
SCHEMBL6469428 0.78 AR (0.58) ARCYP11B2CYP11B1CCNCCDK8
SCHEMBL5368784 0.78 AR (0.58) ARCYP11B2CYP11B1CCNCCDK8
SCHEMBL5365931 0.78 AR (0.65) ARCYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed