SCHEMBL5368784

SCHEMBL5368784

Cc1c[nH]nc1Cn1c(C)c(C#N)c(-c2ccc(C#N)cc2)c1C

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.58
CYP11B2 P19099 3/20 0.36
CHEK1 O14757 1/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
GRIA2 P42262 1/20 0.33
GRIA4 P48058 1/20 0.33
SLC11A2 P49281 1/20 0.33
DHODH Q02127 1/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14347749 0.84 AR (0.47) ARCYP11B2CHEK1CCNCCDK8
SCHEMBL14347768 0.84 AR (0.57) ARCYP11B2CCNCCDK8GRIA2
SCHEMBL5362232 0.80 AR (0.61) ARCYP11B2CCNCCDK8GRIA2
SCHEMBL14347772 0.78 AR (0.53) ARCYP11B2CCNCCDK8
SCHEMBL5365892 0.78 AR (0.65) ARCYP11B2CCNCCDK8CYP11B1
SCHEMBL6469428 0.78 AR (0.58) ARCYP11B2CCNCCDK8GRIA2
SCHEMBL5367267 0.78 AR (0.52) ARCYP11B2CCNCCDK8GRIA2
SCHEMBL5362254 0.78 AR (0.60) ARGRIA2GRIA4FNTAFNTB
SCHEMBL6468889 0.77 AR (0.86) ARCYP11B2CCNCCDK8CYP11B1
SCHEMBL5361308 0.77 CYP11B2 (0.41) ARCYP11B2CCNCCDK8FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed