SCHEMBL5366390

SCHEMBL5366390

Cc1cc(C=C2C(=O)Nc3ccc(CCCl)cc32)oc1C

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
RPS6KA3 P51812 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
DYRK1A Q13627 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
THRB P10828 1/20 0.42
ALOX12 P18054 1/20 0.42
RET P07949 5/20 0.41
LRRK2 Q5S007 2/20 0.41
PDPK1 O15530 3/20 0.41
PDGFRB P09619 1/20 0.40
PTPN1 P18031 1/20 0.40
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.39
ALK Q9UM73 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367282 0.85 KMT2A (0.60) ALDH1A1MAPTRPS6KA3MEN1KMT2A
SCHEMBL5373671 0.83 GSK3B (0.44) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL5363472 0.81 PTPN1 (0.48) ALDH1A1MAPTRPS6KA3MEN1KMT2A
SCHEMBL5369248 0.81 RET (0.65) ALDH1A1MAPTRPS6KA3MEN1KMT2A
SCHEMBL5367384 0.80 RPS6KA3 (0.43) ALDH1A1MAPTRPS6KA3MEN1KMT2A
SCHEMBL6830072 0.80 RPS6KA3 (0.62) ALDH1A1MAPTRPS6KA3MEN1KMT2A
SCHEMBL6855418 0.80 RPS6KA3 (0.62) ALDH1A1MAPTRPS6KA3MEN1KMT2A
SCHEMBL7139419 0.79 MEN1 (0.67) MAPTRPS6KA3MEN1KMT2ALMNA
SCHEMBL7137564 0.79 PSEN1 (0.52) MAPTMEN1KMT2ARETLRRK2
SCHEMBL7134047 0.79 PTPN1 (0.48) ALDH1A1RPS6KA3MEN1KMT2ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK ALDH1A1 2044/4885MAPT 3048/4885RPS6KA3 271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.