SCHEMBL5363472

SCHEMBL5363472

CCc1ccc(C=C2C(=O)Nc3ccc(CCCl)cc32)o1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 12/20 0.48
PTPN2 P17706 2/20 0.48
RET P07949 3/20 0.46
ALDH1A1 P00352 2/20 0.44
DYRK1A Q13627 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
THRB P10828 1/20 0.44
ALOX12 P18054 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPT P10636 1/20 0.41
RPS6KA3 P51812 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7134047 0.89 PTPN1 (0.48) PTPN1PTPN2RETALDH1A1DYRK1A
SCHEMBL5367282 0.86 KMT2A (0.60) PTPN1PTPN2RETALDH1A1DYRK1A
SCHEMBL5369248 0.84 RET (0.65) PTPN1PTPN2RETALDH1A1DYRK1A
SCHEMBL5366390 0.81 ALDH1A1 (0.45) PTPN1RETALDH1A1DYRK1AMEN1
SCHEMBL5357851 0.81 RET (0.53) PTPN1PTPN2RETALDH1A1MEN1
SCHEMBL7133824 0.80 PSEN1 (0.52) RETMAPT
SCHEMBL5728121 0.78 POLB (0.69) PTPN1PTPN2ALDH1A1DYRK1AMEN1
SCHEMBL6304861 0.78 POLB (0.69) PTPN1PTPN2ALDH1A1DYRK1AMEN1
SCHEMBL5728117 0.78 POLB (0.69) PTPN1PTPN2ALDH1A1DYRK1AMEN1
SCHEMBL5373780 0.78 EGFR (0.64) RETALDH1A1ALOX12MAPTRPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK PTPN1 882/4885PTPN2 1051/4885RET 283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.