SCHEMBL5366919

SCHEMBL5366919

O=C(NCC1CN(C(=O)OCc2ccc(F)c(C(F)(F)F)c2)CCO1)c1ccc(O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 7/20 0.46
HTR2A P28223 1/20 0.41
ABAT P80404 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
PTPN7 P35236 1/20 0.41
DUSP3 P51452 1/20 0.41
F2 P00734 1/20 0.41
PLG P00747 1/20 0.41
PRSS1 P07477 1/20 0.41
PRSS2 P07478 1/20 0.41
PRSS3 P35030 1/20 0.41
TPSAB1 Q15661 1/20 0.41
TPSD1 Q9BZJ3 1/20 0.41
TPSG1 Q9NRR2 1/20 0.41
HPGD P15428 2/20 0.40
DRD4 P21917 1/20 0.40
GRIN2B Q13224 3/20 0.40
KCNH2 Q12809 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425369 1.00 ENPP2 (0.46) ENPP2HTR2AABATSIGMAR1PTPN7
SCHEMBL14425368 0.90 ENPP2 (0.49) ENPP2HTR2AABATSIGMAR1F2
SCHEMBL5359620 0.90 ENPP2 (0.49) ENPP2HTR2AABATSIGMAR1F2
SCHEMBL5368400 0.88 ENPP2 (0.47) ENPP2HTR2AABATSIGMAR1F2
SCHEMBL14425314 0.86 F2 (0.48) ENPP2SIGMAR1F2PLGPRSS1
SCHEMBL5362085 0.86 F2 (0.48) ENPP2SIGMAR1F2PLGPRSS1
SCHEMBL14425445 0.86 F2 (0.48) ENPP2SIGMAR1F2PLGPRSS1
SCHEMBL5374371 0.85 ENPP2 (0.47) ENPP2HTR2AABATSIGMAR1F2
SCHEMBL14425378 0.85 ENPP2 (0.47) ENPP2HTR2AABATSIGMAR1F2
SCHEMBL5364450 0.84 GRIN2B (0.48) ENPP2HTR2AABATSIGMAR1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed