SCHEMBL5367155

SCHEMBL5367155

CCOc1cc(C=C2C(=O)Nc3ccc(S(=O)(=O)NC)cc32)ccc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 2/20 0.52
PIM1 P11309 2/20 0.49
PIM3 Q86V86 2/20 0.49
PIM2 Q9P1W9 2/20 0.49
SRC P12931 4/20 0.48
CDK2 P24941 2/20 0.47
DYRK1A Q13627 1/20 0.47
DYRK2 Q92630 1/20 0.47
NTRK1 P04629 1/20 0.47
FCER2 P06734 1/20 0.47
SYK P43405 1/20 0.47
NTRK3 Q16288 1/20 0.47
NTRK2 Q16620 1/20 0.47
PTGS2 P35354 1/20 0.47
KMT2A Q03164 4/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
PLK4 O00444 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362923 0.89 PSEN1 (0.54) NOX4SRCCDK2NTRK1FCER2
SCHEMBL7140878 0.85 SYK (0.55) SRCCDK2NTRK1FCER2SYK
SCHEMBL5376985 0.84 MGAT2 (0.51) NOX4PIM1PIM3PIM2DYRK1A
SCHEMBL5363044 0.84 SRC (0.53) NOX4SRCCDK2NTRK1FCER2
SCHEMBL7139502 0.83 NOX4 (0.54) NOX4SRCCDK2NTRK1FCER2
SCHEMBL5358229 0.83 LRRK2 (0.64) NOX4PIM1PIM3PIM2SRC
SCHEMBL5377083 0.82 SYK (0.50) SRCCDK2NTRK1FCER2SYK
SCHEMBL5359504 0.82 PSEN1 (0.56) NOX4SRCCDK2NTRK1FCER2
SCHEMBL7138006 0.81 SRC (0.57) SRCCDK2NTRK1FCER2SYK
SCHEMBL5365190 0.81 PSEN1 (0.60) SRCCDK2MAPTPLK4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK NOX4 3452/4885PIM1 397/4885PIM3 449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.