SCHEMBL5367296

SCHEMBL5367296

O=C(NCC1CN(C(=O)OCc2ccccc2)CCO1)c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 7/20 0.51
CYP2D6 P10635 4/20 0.51
CYP2C9 P11712 4/20 0.51
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
USP30 Q70CQ3 1/20 0.47
CYP3A4 P08684 3/20 0.46
ENPP2 Q13822 2/20 0.45
HPGD P15428 1/20 0.45
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
TPSAB1 Q15661 1/20 0.43
TPSD1 Q9BZJ3 1/20 0.43
TPSG1 Q9NRR2 1/20 0.43
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425431 0.90 ENPP2 (0.47) GRIN2BCYP2D6CYP2C9MEN1KMT2A
SCHEMBL5359093 0.90 ENPP2 (0.47) GRIN2BCYP2D6CYP2C9MEN1KMT2A
SCHEMBL14425436 0.90 MEN1 (0.50) GRIN2BMEN1KMT2ANPSR1USP30
SCHEMBL14425317 0.90 MEN1 (0.50) GRIN2BMEN1KMT2ANPSR1USP30
SCHEMBL5368740 0.90 MEN1 (0.50) GRIN2BMEN1KMT2ANPSR1USP30
SCHEMBL5371131 0.87 NPC1L1 (0.51) GRIN2BCYP2D6CYP2C9MEN1KMT2A
SCHEMBL5362334 0.86 ENPP2 (0.47) GRIN2BMEN1KMT2ANPSR1USP30
SCHEMBL5369961 0.86 MEN1 (0.46) GRIN2BMEN1KMT2ANPSR1USP30
SCHEMBL5368831 0.85 GRIN2B (0.45) GRIN2BCYP2D6CYP2C9MEN1KMT2A
SCHEMBL14425443 0.85 ENPP2 (0.46) GRIN2BCYP2D6CYP2C9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed