SCHEMBL5368307

SCHEMBL5368307

NC(Cc1cc(F)cc(F)c1)C(O)CNCc1cccc(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.48
CTSD P07339 4/20 0.48
BCHE P06276 1/20 0.39
CTSB P07858 1/20 0.39
BACE2 Q9Y5Z0 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3354961 1.00 BACE1 (0.48) BACE1CTSDBCHECTSBBACE2
SCHEMBL3178597 1.00 BACE1 (0.48) BACE1CTSDBCHECTSBBACE2
SCHEMBL3351909 0.90 BACE1 (0.52) BACE1CTSDCTSBBACE2
SCHEMBL4041091 0.87 BCHE (0.51) BACE1BCHECYP1A2CYP2D6CYP2C19
SCHEMBL3357034 0.86 BCHE (0.49) BACE1CTSDBCHEBACE2
SCHEMBL2874563 0.85 BACE1 (0.53) BACE1CTSDCTSB
SCHEMBL3352827 0.85 BACE1 (0.57) BACE1CTSDCTSBBACE2
SCHEMBL3349064 0.85 BACE1 (0.53) BACE1CTSDCTSB
SCHEMBL3348880 0.85 LMNA (0.50) BACE1CTSDCTSBCYP1A2CYP2D6
SCHEMBL3356792 0.85 BACE1 (0.59) BACE1CTSDCTSBBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565443-A4 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES ELAN PHARM INC (US) 2007-07-18 EP disclosed
EP-1565443-A2 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES Elan Pharmaceuticals, Inc. (US) 2005-08-24 EP disclosed
WO-2004024081-A2 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES ELAN PHARMACEUTICALS, INC. (US) 2004-03-25 WO disclosed