SCHEMBL5368936

SCHEMBL5368936

Cc1cc(Cc2ccc(Br)c(Oc3cc(Cl)cc(C#N)c3)c2F)n[nH]c1=O

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.72
CYP2C9 P11712 2/20 0.72
CYP2C19 P33261 1/20 0.72
KCNH2 Q12809 5/20 0.43
CYP2D6 P10635 1/20 0.33
SLC5A2 P31639 1/20 0.33
SLC22A12 Q96S37 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5375519 0.92 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL4274479 0.91 CYP3A4 (0.86) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL5374302 0.88 CYP3A4 (0.64) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2
SCHEMBL5382037 0.86 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19KCNH2CYP2D6
SCHEMBL4274657 0.86 CYP3A4 (0.91) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2
SCHEMBL5668069 0.85 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2
SCHEMBL5374191 0.84 CYP3A4 (0.75) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2
SCHEMBL5376896 0.84 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2
SCHEMBL4272969 0.84 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2
SCHEMBL5368425 0.84 CYP3A4 (0.86) CYP3A4CYP2C9CYP2C19KCNH2SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed