SCHEMBL5368939

SCHEMBL5368939

Cc1ccc(Cc2ccc(=O)[nH]n2)cc1Oc1cccc(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.64
SLC6A4 P31645 3/20 0.39
HTR2A P28223 1/20 0.39
KCNH2 Q12809 1/20 0.39
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
PDE5A O76074 1/20 0.36
PDE9A O76083 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A3 Q01959 2/20 0.36
AKR1B1 P15121 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371174 0.89 CYP3A4 (0.51) CYP3A4PTGS1PTGS2ALDH1A1TSHR
SCHEMBL5365181 0.89 CYP3A4 (0.67) CYP3A4SLC6A4HTR2AKCNH2SLC6A2
SCHEMBL5367092 0.88 CYP3A4 (0.66) CYP3A4SLC6A4HTR2AKCNH2PTGS1
SCHEMBL5370245 0.88 CYP3A4 (0.63) CYP3A4SLC6A4HTR2AKCNH2PTGS1
SCHEMBL5413137 0.88 CYP3A4 (0.50) CYP3A4USP2CYP1A2CYP2C9TSHR
SCHEMBL5377723 0.88 CYP3A4 (0.66) CYP3A4SLC6A4HTR2AKCNH2SLC6A2
SCHEMBL5365171 0.88 CYP3A4 (0.49) CYP3A4SLC6A4HTR2AKCNH2
SCHEMBL5370985 0.88 CYP3A4 (0.48) CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5372601 0.87 CYP3A4 (0.62) CYP3A4SLC6A4HTR2AKCNH2PTGS1
SCHEMBL5370972 0.87 CYP3A4 (0.49) CYP3A4FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed