SCHEMBL5370985

SCHEMBL5370985

Cc1ccc(Cc2ccc(=O)[nH]n2)cc1Oc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.48
DAO P14920 1/20 0.37
TTR P02766 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
THRA P10827 2/20 0.36
THRB P10828 2/20 0.36
BRD4 O60885 1/20 0.36
PARP1 P09874 1/20 0.35
PDE10A Q9Y233 1/20 0.35
SRD5A2 P31213 1/20 0.34
IDH1 O75874 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
S1PR2 O95136 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371174 0.90 CYP3A4 (0.51) CYP3A4TSHRTHRATHRBPARP1
SCHEMBL5413137 0.89 CYP3A4 (0.50) CYP3A4CYP2C9TSHRCYP2C19IDH1
SCHEMBL5365171 0.88 CYP3A4 (0.49) CYP3A4THRATHRB
SCHEMBL5368939 0.88 CYP3A4 (0.64) CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5370972 0.88 CYP3A4 (0.49) CYP3A4THRATHRBPARP1ADORA2A
SCHEMBL5365245 0.88 CYP3A4 (0.49) CYP3A4THRATHRBPARP1ADORA2A
SCHEMBL5370472 0.87 CYP3A4 (0.48) CYP3A4DAOTTRCYP2C9TSHR
SCHEMBL5365424 0.87 CYP3A4 (0.48) CYP3A4TTRCYP2C9TSHRCYP2C19
SCHEMBL4367667 0.85 CYP3A4 (0.53) CYP3A4DAOTTRCYP2C9TSHR
SCHEMBL5368917 0.85 CYP3A4 (0.48) CYP3A4DAOTTRCYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed