SCHEMBL5369110

SCHEMBL5369110

Cc1cc(Cc2ccc(Br)c(Oc3ccccc3)c2)n[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
TSHR P16473 1/20 0.39
BRD4 O60885 2/20 0.39
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PDE10A Q9Y233 1/20 0.35
PARP1 P09874 5/20 0.35
TTR P02766 1/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385763 0.86 CYP3A4 (0.43) DAOCYP3A4CYP2C9CYP2C19TSHR
SCHEMBL5370938 0.86 CYP3A4 (0.38) DAOCYP3A4CYP2C9CYP2C19TSHR
SCHEMBL5385101 0.84 DAO (0.38) DAOCYP3A4CYP2C9CYP2C19TSHR
SCHEMBL5368917 0.82 CYP3A4 (0.48) DAOCYP3A4CYP2C9CYP2C19TSHR
SCHEMBL5365352 0.81 CYP3A4 (0.41) DAOCYP3A4CYP2C9CYP2C19TSHR
SCHEMBL5374033 0.80 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19TSHRPARP1
SCHEMBL5372554 0.78 CYP3A4 (0.44) DAOCYP3A4CYP2C9CYP2C19TSHR
SCHEMBL1194422 0.77 DAO (0.54) DAOCYP2C9TSHRKMT2APARP1
SCHEMBL5373895 0.77 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5368768 0.76 CYP3A4 (0.42) DAOCYP3A4CYP2C9CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed