SCHEMBL5368917

SCHEMBL5368917

O=c1ccc(Cc2ccc(Br)c(Oc3ccccc3)c2)n[nH]1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.48
THRA P10827 2/20 0.41
THRB P10828 2/20 0.41
DAO P14920 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NTRK1 P04629 1/20 0.34
NTRK3 Q16288 1/20 0.34
NTRK2 Q16620 1/20 0.34
AKR1B1 P15121 2/20 0.34
TTR P02766 2/20 0.34
TSHR P16473 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CYP1A2 P05177 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377627 0.88 CYP3A4 (0.64) CYP3A4THRATHRBAKR1B1
SCHEMBL5375017 0.85 CYP3A4 (0.51) CYP3A4THRATHRBDAOAKR1B1
SCHEMBL5370985 0.85 CYP3A4 (0.48) CYP3A4THRATHRBDAOTTR
SCHEMBL4367667 0.85 CYP3A4 (0.53) CYP3A4THRATHRBDAOMEN1
SCHEMBL5370328 0.85 CYP3A4 (0.47) CYP3A4THRATHRB
SCHEMBL5370472 0.84 CYP3A4 (0.48) CYP3A4THRATHRBDAOMEN1
SCHEMBL5365424 0.84 CYP3A4 (0.48) CYP3A4TTRTSHRCYP2C9CYP2C19
SCHEMBL5369110 0.82 DAO (0.39) CYP3A4THRATHRBDAOMEN1
SCHEMBL5366909 0.82 CYP3A4 (0.46) CYP3A4THRATHRBDAONTRK1
SCHEMBL5377193 0.81 CYP3A4 (0.50) CYP3A4DAOAKR1B1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed