SCHEMBL5369145

SCHEMBL5369145

O=c1ccc(Cc2ccc(Cl)c(Oc3ccc(Cl)cc3Cl)c2)n[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.48
TTR P02766 4/20 0.42
FFAR1 O14842 2/20 0.40
AKR1B1 P15121 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
PGR P06401 1/20 0.38
HSP90AA1 P07900 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
MAPT P10636 1/20 0.38
HSPA5 P11021 1/20 0.38
HPGD P15428 1/20 0.38
CBR1 P16152 1/20 0.38
TBXA2R P21731 1/20 0.38
AGTR1 P30556 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5369034 0.94 CYP3A4 (0.50) CYP3A4TTRAKR1B1KMT2ALMNA
SCHEMBL5374337 0.88 CYP3A4 (0.47) CYP3A4AKR1B1SLC6A2SLC6A3SLC6A4
SCHEMBL5374390 0.87 CYP3A4 (0.46) CYP3A4AKR1B1KMT2ALMNA
SCHEMBL5373719 0.87 CYP3A4 (0.46) CYP3A4TTRAKR1B1LMNASLC6A4
SCHEMBL5373613 0.87 CYP3A4 (0.51) CYP3A4FFAR1AKR1B1LMNASLC6A4
SCHEMBL5377021 0.85 AR (0.41) CYP3A4FFAR1SLC6A3SLC6A4
SCHEMBL5370291 0.85 CYP3A4 (0.43) CYP3A4AKR1B1SLC6A2LMNAMAPT
SCHEMBL5368714 0.84 CYP3A4 (0.53) CYP3A4FFAR1AKR1B1KMT2AMAPT
SCHEMBL5365181 0.84 CYP3A4 (0.67) CYP3A4AKR1B1SLC6A2SLC6A3SLC6A4
SCHEMBL4367667 0.82 CYP3A4 (0.53) CYP3A4TTRAKR1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed