SCHEMBL5374337

SCHEMBL5374337

O=c1ccc(Cc2ccc(Cl)c(Oc3ccccc3Cl)c2)n[nH]1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.47
AKR1B1 P15121 4/20 0.37
CAMK2A Q9UQM7 1/20 0.37
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
CXCL8 P10145 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377719 0.91 CYP3A4 (0.46) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5367073 0.91 CYP3A4 (0.44) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5373947 0.91 CYP3A4 (0.44) CYP3A4AKR1B1PRMT5WDR77CYP2C9
SCHEMBL5374344 0.90 CYP3A4 (0.43) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5373451 0.89 CYP3A4 (0.48) CYP3A4AKR1B1CAMK2A
SCHEMBL4367667 0.89 CYP3A4 (0.53) CYP3A4AKR1B1CYP2C9TSHRCYP2C19
SCHEMBL5369034 0.89 CYP3A4 (0.50) CYP3A4AKR1B1
SCHEMBL5369145 0.88 CYP3A4 (0.48) CYP3A4AKR1B1SLC6A2SLC6A4SLC6A3
SCHEMBL5374946 0.88 CYP3A4 (0.42) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5382509 0.88 CYP3A4 (0.42) CYP3A4PRMT5WDR77FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed