SCHEMBL5370073

SCHEMBL5370073

Cc1cccc2c(=O)[nH]cnc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 1.00
PIM1 P11309 2/20 0.64
RPS6KA3 P51812 2/20 0.64
AURKA O14965 1/20 0.64
DAPK3 O43293 1/20 0.64
JAK2 O60674 1/20 0.64
PRKD3 O94806 1/20 0.64
MAP4K4 O95819 1/20 0.64
PAK4 O96013 1/20 0.64
ABL1 P00519 1/20 0.64
CSF1R P07333 1/20 0.64
RET P07949 1/20 0.64
IGF1R P08069 1/20 0.64
MET P08581 1/20 0.64
PDGFRB P09619 1/20 0.64
FGFR1 P11362 1/20 0.64
PDGFRA P16234 1/20 0.64
PRKACA P17612 1/20 0.64
FLT1 P17948 1/20 0.64
LTK P29376 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29443212 1.00 PARP1 (1.00) PARP1PIM1RPS6KA3AURKADAPK3
Trifluoroacetic Acid SCHEMBL31483798 0.87 PARP1 (0.75) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL12068009 0.79 PARP1 (0.66) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL16006387 0.79 PARP1 (0.65) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL1387233 0.78 PARP1 (0.64) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL2447579 0.78 PARP1 (1.00) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL526730 0.78 PARP1 (1.00) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL21895445 0.78 PARP1 (1.00) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL20435416 0.78 PARP1 (0.64) PARP1PIM1RPS6KA3AURKADAPK3
SCHEMBL16097896 0.78 PARP1 (0.64) PARP1PIM1RPS6KA3AURKADAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 137 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106086956-B Alkaline non-cyanide electrodepositing zinc-nickel alloy additive and its application 哈尔滨工业大学 2019-03-01 CN claimed
CN-106086956-A Alkaline non-cyanide electrodepositing zinc-nickel alloy additive and application thereof 哈尔滨工业大学 2016-11-09 CN claimed
US-20250059157-A1 TLR7/8 ANTAGONISTS AND USES THEREOF MERCK PATENT GMBH (DE) 2025-02-20 US disclosed
US-12030858-B2 PARP inhibitors for treating cancer and asthma OREGON HEALTH & SCIENCE UNIVERSITY (US) 2024-07-09 US disclosed
EP-3889145-B1 8-CYANO-5-PIPERIDINO-QUINOLINES AS TLR7/8 ANTAGONISTS AND THEIR USES FOR TREATING IMMUNE DISORDERS MERCK PATENT GMBH (DE) 2024-02-21 EP disclosed
WO-2023217906-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2023-11-16 WO disclosed
US-20230303514-A1 TLR7/8 ANTAGONISTS AND USES THEREOF MERCK PATENT GMBH (DE) 2023-09-28 US disclosed
CN-116804001-A Quinazolinone derivative containing pyridinium and preparation method and application thereof 江苏海洋大学 2023-09-26 CN disclosed
US-11739071-B2 Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors VALO HEALTH, INC. (US) 2023-08-29 US disclosed
US-11739071-B2 Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors VALO HEALTH, INC. (US) 2023-08-29 US disclosed
US-11739071-B2 Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors VALO HEALTH, INC. (US) 2023-08-29 US disclosed
US-7217737-B2 Method and compositions for inhibiting cell proliferative disorders YISSUM RESEARCH AND DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2007-05-15 US disclosed
US-20040242684-A1 Method and compositions for inhibiting cell proliferative disorders YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM 2004-12-02 US disclosed
US-6596878-B2 Protein kinase inhibitor compositio; used to treat cell proliferative disorders such as cancers charcterized by over-activity or inappropriate activity HER2 or EGFR. YISSUM RESEARCH & DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY (IL) 2003-07-22 US disclosed
US-20020068687-A1 Methods and compositions for inhibiting cell proliferative disorders CHEN HUI (US) 2002-06-06 US disclosed
US-5789427-A ANTITUMOR, ANTICANCER AGENTS SUGEN, INC. (US) 1998-08-04 US disclosed
US-5773476-A KINASE INHIBITORS SUGEN, INC. (IL) 1998-06-30 US disclosed
WO-1995024190-A2 RECEPTOR TYROSINE KINASE INHIBITORS FOR INHIBITING CELL PROLIFERATIVE DISORDERS AND COMPOSITIONS THEREOF SUGEN, INC. (US) 1995-09-14 WO disclosed
US-5401745-A Cardiovascular disorders or hypotensive agents MERCK & CO., INC. (US) 1995-03-28 US disclosed
WO-1994021259-A1 QUINAZOLINONES SUBSTITUTED WITH PHENOXYPHENYLACETIC ACID DERIVATIVES MERCK & CO., INC. (US) 1994-09-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303514-A1 TLR7/8 ANTAGONISTS AND USES THEREOF TLR7, TLR8, TLR9 PARP1 866/4885PIM1 3665/4885RPS6KA3 1953/4885
US-11739071-B2 Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors USP7, UBQLN1, UBA7 PARP1 997/4885PIM1 3951/4885RPS6KA3 856/4885
US-20040242684-A1 Method and compositions for inhibiting cell proliferative disorders ERBB2, EGFR, MKI67 PARP1 856/4885PIM1 583/4885RPS6KA3 400/4885
US-12030858-B2 PARP inhibitors for treating cancer and asthma PARP1, PARP2, PARP11 PARP1 1/4885PIM1 652/4885RPS6KA3 943/4885
US-20250059157-A1 TLR7/8 ANTAGONISTS AND USES THEREOF TLR7, TLR8, TLR9 PARP1 866/4885PIM1 3665/4885RPS6KA3 1953/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.