SCHEMBL5370974

SCHEMBL5370974

Cc1cc(Cc2ccc(Cl)c(Oc3cc(Cl)cc(Cl)c3)c2F)n[nH]c1=O

nearest known ligand 0.73

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.73
CYP2C9 P11712 1/20 0.73
CYP2C19 P33261 1/20 0.73
SLC5A2 P31639 1/20 0.41
HTR2A P28223 3/20 0.34
SLC6A4 P31645 3/20 0.34
KCNH2 Q12809 3/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PARP1 P09874 1/20 0.31
P2RX7 Q99572 5/20 0.31
DRD1 P21728 1/20 0.31
POLB P06746 1/20 0.30
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4274479 0.91 CYP3A4 (0.86) CYP3A4CYP2C9CYP2C19SLC5A2HTR2A
SCHEMBL5368877 0.89 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19SLC5A2LMNA
SCHEMBL4274657 0.87 CYP3A4 (0.91) CYP3A4CYP2C9CYP2C19SLC5A2HTR2A
SCHEMBL4272969 0.85 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5368425 0.85 CYP3A4 (0.86) CYP3A4CYP2C9CYP2C19SLC5A2HTR2A
SCHEMBL5377687 0.84 CYP3A4 (0.64) CYP3A4CYP2C9CYP2C19SLC5A2
SCHEMBL5375519 0.83 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19SLC5A2HTR2A
SCHEMBL4278760 0.83 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19SLC5A2
SCHEMBL5368624 0.83 CYP3A4 (0.80) CYP3A4CYP2C9CYP2C19SLC5A2HTR2A
SCHEMBL5344677 0.82 CYP3A4 (0.81) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed