SCHEMBL5371308

SCHEMBL5371308

CCc1cccc(CNC[C@@H](O)[C@H](Cc2cc(F)cc(F)c2)N(C(=O)CN)C(=O)c2ccc(Cl)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.50
CTSD P07339 4/20 0.50
CTSB P07858 12/20 0.46
BACE2 Q9Y5Z0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5372922 0.92 BACE1 (0.49) BACE1CTSDCTSBBACE2
SCHEMBL5375804 0.90 BACE1 (0.52) BACE1CTSDCTSBBACE2
SCHEMBL5374086 0.89 BACE1 (0.49) BACE1CTSDCTSBBACE2
SCHEMBL6699273 0.82 BACE1 (0.49) BACE1CTSDCTSBBACE2
SCHEMBL3490928 0.82 BACE1 (0.47) BACE1CTSDCTSB
SCHEMBL3490933 0.82 BACE1 (0.47) BACE1CTSDCTSB
SCHEMBL6697214 0.81 BACE1 (0.46) BACE1CTSDCTSBBACE2
SCHEMBL3490931 0.78 BACE1 (0.48) BACE1CTSDCTSB
SCHEMBL6697182 0.78 BACE1 (0.49) BACE1CTSDCTSB
SCHEMBL3490123 0.77 BACE1 (0.49) BACE1CTSDCTSBBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed