SCHEMBL5375804

SCHEMBL5375804

CCc1cccc(CNC[C@@H](O)[C@H](Cc2cc(F)cc(F)c2)N(C(=O)CN)C(=O)c2ccc(C(C)(C)C)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.52
CTSD P07339 4/20 0.49
CTSB P07858 11/20 0.46
BCHE P06276 1/20 0.41
BACE2 Q9Y5Z0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371308 0.90 BACE1 (0.50) BACE1CTSDCTSBBACE2
SCHEMBL5372922 0.87 BACE1 (0.49) BACE1CTSDCTSBBACE2
SCHEMBL6699273 0.81 BACE1 (0.49) BACE1CTSDCTSBBACE2
SCHEMBL6697182 0.80 BACE1 (0.49) BACE1CTSDCTSB
SCHEMBL6697214 0.80 BACE1 (0.46) BACE1CTSDCTSBBACE2
SCHEMBL5374086 0.80 BACE1 (0.49) BACE1CTSDCTSBBACE2
SCHEMBL5377569 0.79 BACE1 (0.53) BACE1CTSDCTSBBCHEBACE2
SCHEMBL5375739 0.77 BACE1 (0.54) BACE1CTSDCTSB
SCHEMBL3355547 0.75 BACE1 (0.65) BACE1CTSDCTSBBCHE
SCHEMBL13308177 0.75 BACE1 (0.65) BACE1CTSDCTSBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed