SCHEMBL5372848

SCHEMBL5372848

N#Cc1cc(C#N)cc(Oc2cccc(Cc3ccc(=O)[nH]n3)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.45
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
KCNH2 Q12809 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
HRH3 Q9Y5N1 1/20 0.33
MMP13 P45452 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366793 0.88 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19MMP13
SCHEMBL5377193 0.84 CYP3A4 (0.50) CYP3A4CYP2C9CYP2C19PARP1
SCHEMBL5377482 0.82 CYP3A4 (0.57) CYP3A4PRMT5WDR77THRATHRB
SCHEMBL5377805 0.81 CYP3A4 (0.45) CYP3A4KCNH2CYP2C9CYP2C19CYP11B1
SCHEMBL14570721 0.81 CYP3A4 (0.41) CYP3A4KCNH2CYP2C9CYP2C19THRA
SCHEMBL5377579 0.81 CYP3A4 (0.52) CYP3A4PRMT5WDR77KCNH2CYP2C9
SCHEMBL5374410 0.81 CYP3A4 (0.49) CYP3A4PRMT5WDR77PARP1
SCHEMBL5370328 0.81 CYP3A4 (0.47) CYP3A4PRMT5WDR77THRATHRB
SCHEMBL5375295 0.81 CYP3A4 (0.47) CYP3A4PRMT5WDR77CYP2C9CYP2C19
SCHEMBL5369070 0.81 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed